GeneTex is committed to establishing the most extensive product line of recombinant monoclonal antibodies for human GPCRs. These antibodies will be thoroughly characterized through enhanced “Five Pillar” validation strategies that feature knockdown/knockout lysates, comparable antibodies, cell fractionation, detection of endogenous GPCR expression, and overexpression. In addition, specialized testing using human GPCR arrays will be utilized when feasible. The goal is to generate the most diverse, expansive, and meticulously verified antibody reagents for GPCR biology research.

 

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Explore Our GPCR Antibodies

 

 

Class A

 

Subclass

Target

5-hydroxytryptamine

5-hydroxytryptamine Receptor 7 (HTR7)
5-hydroxytryptamine 5-hydroxytryptamine Receptor 1E (5-HT1E)

Acetylcholine

Cholinergic Receptor Muscarinic 1 (mAChR M1)

Adenosine

Adenosine A1 Receptor (ADORA1)

Adrenoceptors

Alpha 1a Adrenergic Receptor (ADRA1A)

Adrenoceptors Alpha 1d Adrenergic Receptor (ADRA1D)
Adrenoceptors Alpha 2a Adrenergic Receptor (ADRA2A)
Adrenoceptors Beta 1 Adrenergic Receptor (ADRB1)

Adrenoceptors

Beta 2 Adrenergic Receptor (ADRB2)

Angiotensin Angiotensin II Receptor Type 1 (AGTR1)
Apelin Apelin Receptor (APLNR)
Cannabinoid Cannabinoid Receptor 2 (CNR2)
Chemokine C-C Motif Chemokine Receptor 1 (CCR1)
Chemokine C-C Motif Chemokine Receptor 2 (CCR2)
Chemokine C-C Motif Chemokine Receptor 4 (CCR4)
Chemokine C-C Motif Chemokine Receptor 5 (CCR5)
Chemokine C-C Motif Chemokine Receptor 7 (CCR7)
Chemokine C-C Motif Chemokine Receptor 9 (CCR9)
Chemokine C-C Motif Chemokine Receptor 10 (CCR10)
Chemokine Atypical Chemokine Receptor 4 (CCR11)
Chemokine C-X-C Motif Chemokine Receptor 1 (CXCR1)
Chemokine C-X-C Motif Chemokine Receptor 2 (CXCR2)
Chemokine C-X-C Motif Chemokine Receptor 3 (CXCR3)
Chemokine C-X-C Motif Chemokine Receptor 4 (CXCR4)
Chemokine C-X-C Motif Chemokine Receptor 5 (CXCR5)
Chemokine C-X-C Motif Chemokine Receptor 6 (CXCR6)
Chemokine Atypical Chemokine Receptor 3 (CXCR7)
Class A Orphans Leucine Rich Repeat Containing G Protein-Coupled Receptor 6 (LGR6)
Complement Complement C3A Receptor 1 (C3AR1)
Dopamine Dopamine Receptor D1 (DRD1)
Dopamine Dopamine Receptor D2 (DRD2)
Dopamine Dopamine Receptor D4 (DRD4)
Dopamine Dopamine Receptor D5 (DRD5)
Endothelin Endothelin Receptor Type B (Ednrb)
Formylpeptide Formyl Peptide Receptor 2 (FPRL1)

Free fatty acid

Free Fatty Acid Receptor 1 (GPR40)

Free fatty acid Free Fatty Acid Receptor 2 (GPR43)
Free fatty acid Free Fatty Acid Receptor 4 (GPR120)
Glycoprotein Follicle Stimulating Hormone Receptor (FSHR)

Glycoprotein

Thyroid Stimulating Hormone Receptor (TSHR)

Gonadotrophin Gonadotropin Releasing Hormone Receptor (GnRHR)
Histamine Histamine Receptor H1 (HRH1)

Lysophospholipid

Lysophosphatidic Acid Receptor 2 (EDG-4/LPAR2)
Lysophospholipid PAF Receptor (PTAFR)
Lysophospholipid Sphingosine-1-phosphate Receptor 2 (S1PR2)
Melanocortin Melanocortin 1 Receptor (MC1R)
Melanocortin Melanocortin 4 Receptor (MC4R)
Melanocortin Melanocortin 5 Receptor (MC5R)
Opioid Opioid Receptor Delta 1 (OPRD1)
Opioid Opioid Receptor Mu 1 (OPRM1)
Opsins Opsin Red / Green (OPN1MW2)
Opsins Retinal G Protein Coupled Receptor (RGR)
Opsins Rhodopsin (RHO)
Prostanoid Prostaglandin E Receptor 3 (PTGER3)
P2Y Purinergic Receptor P2Y1 (P2Y1)
P2Y Purinergic Receptor P2Y2 (P2Y2)
P2Y Purinergic Receptor P2Y11 (P2Y11)
P2Y Purinergic Receptor P2Y12 (P2Y12)
Somatostatin Somatostatin Receptor 2 (SSTR2)
Somatostatin Somatostatin Receptor 3 (SSTR3)
Somatostatin Somatostatin Receptor 4 (SSTR4)
Somatostatin Somatostatin Receptor 5 (SSTR5)
Tachykinin Neurokinin 1 Receptor (NK1R)

 

 

 

Class B1

 

Subclass

Target

Calcitonin

Calcitonin Receptor Like Receptor (CRLR)

Glucagon family

Glucagon Like Peptide 1 Receptor (GLP1R)

Parathyroid

Parathyroid Hormone 1 Receptor (PTH1R)

VIP and PACAP

Vasoactive Intestinal Peptide Receptor 2 (VPAC2)

 

Class B2

 

Subclass

Target

Adhesion

Adhesion G Protein-Coupled Receptor B2 (BAI2)

Adhesion

Adhesion G Protein-Coupled Receptor B3 (BAI3)

Adhesion

Adhesion G Protein-Coupled Receptor E5 (CD97)

Adhesion

Adhesion G Protein-Coupled Receptor G3 (GPR97)

Adhesion Adhesion G Protein-Coupled Receptor G5 (GPR114)

 

Class C

 

Subclass

Target

Calcium-sensing

Calcium Sensing Receptor (CASR)

Class C Orphans G Protein-Coupled Receptor Class C Group 5 Member A (GPRC5A)

Class C Orphans

G protein-Coupled Receptor Class C Group 5 Member C (GPRC5C)

Class C Orphans

G protein-Coupled Receptor Class C Group 5 Member D (GPRC5D)
GABA Gamma-aminobutyric Acid Type B Receptor Subunit 1 (GABBR1)

Metabotropic glutamate

Glutamate Metabotropic Receptor 4 (mGluR4)
Metabotropic
glutamate
Glutamate Metabotropic Receptor 5 (mGluR5)

 

Class F

 

Subclass

Target

Frizzled

Frizzled 4 (FZD4)

Frizzled

Frizzled 9 (FZD9)

Frizzled Smoothened Homolog (SMO)

 

 

Class Taste 2

 

Subclass

Target

Taste 2

Taste 2 Receptor Member 38 (TAS2R38)

 

 

 

 

 

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